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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T17284 | Zardaverine | BY 290,B 84290 | PDE |
Zardaverine (BY 290) is an orally available, selective and potent PDE3/4 inhibitor with bronchodilator activity and anti-hepatocarcinogenic activity.Zardaverine's action in platelets is mediated by PDE III isoenzymes and... | |||
T12407 | Pepstatin Ammonium | Pepstatin A Ammonium | Others |
Pepstatin Ammonium is a specific inhibitor of aspartic proteaseproduced by actinomycetes(hemoglobin-pepsin, hemoglobin-proctase, casein-pepsin, casein-proctase, casein-acid protease and hemoglobin-acid protease with IC50... | |||
T82514 | EAC3I | ||
EAC3I, an autocamtide-3 derived inhibitory peptide with the sequence KKALHRQEAVDAL, is a bioactive peptide that mimics the autoinhibitory region of the CaMKII regulatory domain (residues 278–290). It functions by competi... | |||
T75705 | Pepstatin Trifluoroacetate | ||
Pepstatin Trifluoroacetate (Pepstatin A), a specific and orally active aspartic protease inhibitor produced by actinomycetes, demonstrates inhibition efficacy with IC50 values of 4.5 nM, 6.2 nM, 150 nM, 290 nM, 520 nM, a... | |||
TN4140 | Glochidiol | Others | |
Glochidiol exhibits strong inhibitory effects against all three human tumor cell lines (MCF-7, NCI-H-460 and SF-268), it exerts its antiproliferative activity through the involvement of apoptosis. It exhibits a strong in... |